What is the purpose of the Cataladon: instruction and feedback

Cathadolone is an analgesic drug of a non-opioid pharmacological group.

The main active ingredient is flupirtine, which has an analgesic effect of the central action, since it is able to selectively activate the neuronal channels of potassium nature. In addition, the drug may have a minor miorelaxing and neurotrophic pharmacological action.

On this page you will find all information about Cathadolone: the full instructions for use on this medication, average prices in pharmacies, complete and incomplete analogs of the drug, as well as reviews of people who have already used Catadolone. Want to leave your opinion? Please write in the comments.

Clinical and pharmacological group

A non-opioid analgesic of central action.

Conditions of leave from pharmacies

It is released on prescription.

Price list

How much does the Catadolon cost? The average price in pharmacies is at the level of500 rubles.

Form of issue and composition

The cadadolon is available in the form of capsules for oral administration in blister packs of 10 pieces for 1, 3 or 5 blisters in a carton.

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Active ingredient: one capsule contains 100 mg of flupirtine maleate.
Auxiliary components: calcium hydrophosphate dihydrate, copovidone, magnesium stearate, colloidal silicon dioxide, gelatin, purified water, E 171 and E 172 dyes, sodium lauryl sulfate.

Pharmacological effect

Medication Catadolon has analgesic effect and refers to non-opioid analgesics of central action. The main substance in the capsules flupirtine - refers to the selective activators of neutral potassium channels. When taking a therapeutic dose, the drug does not bind to adrenoreceptors and cholinergic receptors.

Due to this action the drug has a pronounced analgesic property. In the process of selective opening of neutral potassium channels with a joint release of potassium ions, the resting level of the neuron is normalized. It becomes less irritable and painful. Cagedolone tablets in a short time relieve the patient of mild to moderate pain. Also, the drug has a muscle relaxant effect.

Indications for use

When appoint? Indication for the use of Catadolone is the presence of pain syndrome of various etiologies, namely:

Violations of the menstrual cycle with painful phenomena.
Post-traumatic neuropathic pain.
Painful muscle spasm, including fibromyalgia.
Tension headaches.
Oncopathology with pain syndrome.
Postoperative period.

Contraindications

You can not prescribe medicine for the following pathologies and diseases:

liver disease;
children under 18;
chronic alcoholism;
patients who have a history of propensity to develop renal encephalopathy;
when taken together with drugs, which have a hepatotoxic effect;
recently cured ringing in the ears;
increased sensitivity to the main substance or its components;
with caution is prescribed by doctors to the elderly.

During the treatment period, the vehicle should try to avoid driving and managing precise mechanisms.

Application in pregnancy and lactation

Although no damaging effect on the fetus has been detected so far, but in accordance with the currently valid general provision on the use of medicines Catadolone is not recommended for pregnant women. Until now, clinical experience has not been accumulated with the use of the drug in pregnant women.

If, in the case of an urgent testimony to the puerpera, it is necessary to appoint Cathadolone, then this is done provided that breastfeeding ceases for the duration of treatment. In studies conducted so far, it was found that the active substance in small amounts penetrates into the mother's milk.

Instructions for use

The instructions for use indicate that the Catadolone is taken internally.

The capsule should be swallowed whole, without chewing and washing down with a sufficient amount of liquid (preferably water). If possible, the drug should be taken while in a vertical position. In exceptional cases, the capsule of the drug Catadolone can be opened and taken inside / through the probe only the contents of the capsule.

When ingestion of the contents of the capsule, it is recommended to neutralize its bitter taste by eating food, for example, a banana.

The recommended dose of the drug is 100 mg (1 caps.) 3-4 times / day, if possible, with equal intervals between doses. At the expressed pains - on 200 mg (2 caps.) 3 times / sut. The maximum daily dose is 600 mg (6 caps.).
The dose is selected depending on the intensity of pain and individual sensitivity to the drug. Use the minimum effective dose for the shortest possible time. Duration of treatment should not exceed 2 weeks.
Older patients (over 65 years) at the beginning of treatment are prescribed 100 mg (1 caps.) 2 times / day, morning and evening.

In patients with renal insufficiency, the concentration of creatinine in the blood plasma should be monitored. The maximum daily dose should not exceed 300 mg (3 caps.). In patients with mild to moderate renal failure, dose adjustment is not required. In patients with severe renal insufficiency or hypoalbuminemia, the maximum daily dose should not exceed 300 mg (3 caps.).

If it is necessary to prescribe the drug at higher doses, careful monitoring is established for the patients.

Side effects

When taking the drug, the following side effects are possible:

Subcutaneous tissues and skin: sweating.
Depression, sleep disturbance, tremor, headache, nervousness and / or restlessness, dizziness, confused consciousness - CNS.
Bile ducts and liver: an increase in the activity of liver enzymes, hepatic insufficiency, hepatitis.
Body of vision: impaired vision.
GI tract: pain in the stomach, flatulence, constipation, indigestion, abdominal pain, bouts of nausea, dryness of the oral mucosa, vomiting, diarrhea.
Other: deterioration or lack of appetite, weakness and / or fatigue (in 15% of patients), especially at the beginning of therapy.
Immune system: infrequently - allergic manifestations (skin rashes, fever, itching, hives), hypersensitivity to the drug.

As a rule, adverse reactions depend on the dose of Catadolone (with the exception of allergic manifestations). After the completion of therapy, they disappear on their own.

Overdose

There is confusion, tachycardia, nausea, dryness of the mucous membranes. In case of an overdose - gastric lavage and treatment, according to the manifested symptoms.

special instructions

At the age of 65 years and older, with expressed signs of hepatic and / or renal insufficiency, and also with hypoalbuminemia, dose adjustment is required.
In patients with reduced renal or hepatic function, it is necessary to control the creatinine content in the urine and the activity of liver enzymes.
The use of the drug in high doses in certain cases can cause the urine to turn green, which is not a clinical sign of any disease.
When flupirtine is used, false positive tests for bilirubin, protein in the urine and urobilinogen are possible. A similar reaction can be in the quantitative determination of the level of bilirubin in the blood plasma.

Given the ability of the Catadolone to weaken attention and slow the reaction rate, during treatment it is recommended refrain from driving transport and practicing potentially hazardous activities.

Drug Interactions

When prescribing the drug Kataladon with diazepam or warfarin, it is possible to enhance the therapeutic effect of the latter.

When used in parallel with the preparation of coumarin derivatives, the prothrombin index should be constantly monitored by patients. If necessary, the dose of coumarin is adjusted.

With the simultaneous administration of the drug Kadadolon with muscle relaxants or sedatives, the therapeutic the effect of the latter, which should be taken into account and select the dose correctly, so that the patient does not develop signs of an overdose.

It is not recommended to combine this drug with paracetamol derivatives, since in this case the risk of toxic damage to the liver increases.

Reviews

We picked up some of the people's comments about the Catadolon drug:

Marina. At me a problem with a neck, very often happens, that can zaklinit and zaschimit a nerve. The pain is unbearable. The neurologist prescribed Catadolone. The first time took him about 3 months ago, drank 3 days, everything went away. Yesterday the same thing happened again, I decided to take these pills (I take 2 capsules 2 times a day, as the doctor prescribed). Half an hour later, a wild dizziness began, my eyesight grew turbid, my hands began to tremble tremendously. All has passed or has taken place in current of 1-2 hours, the pain in a neck too became noticeably less. I wrote off everything that I drank a glass of wine the night before. Today I woke up and decided to repeat the experiment. The result: there is no dizziness, there is general weakness and shaking hands. The first time the capsules were taken 3 months ago, nothing of the kind happened.
Natalia. I katadolon great help with pain in the spine and with toothache. At one time, many painkillers were tried, but none of my body was suitable. Native, for example, helps the ketans - I do not. Some kind of special sensitivity to many drugs. And the catadolon coped with the pain. Now I always carry it with me in my purse just in case and at home in the medicine cabinet always lies. Of course, it would be better to dispense with drugs, but when there is pain there is nothing else left.
Irina. At me a congenital anomaly of a backbone - an additional vertebra in a waist. I went for a drive on skis - fell, pinched a nerve, gave in a leg. In general, I was so blind that I could not reach the toilet. The blockades with novocaine did not help at all. The nurse pityed me, gave 100 mg of cadetolon, and the second, she said to drink in the evening. After the second pill I got up the next day, and before that lay a week. I went to work. Since then, more than 10 years have passed, the back does not bother anymore.