To relax the muscles, the muscle relaxants

Muscle relaxants

Muscle relaxation products are organic compounds, the molecule of which contains 2 quaternary nitrogen atoms.

Initially, to achieve this effect, plants grown in South America were used, later they began to manufacture synthetic drugs to relax the muscles.

This led to the development of anesthesiology and surgery. In the article we will tell you what medicines are available to relax the muscles.

Another important property of muscle relaxants is the effective protection of a person from stress during surgery. It is provided by the blocking of neuromuscular transmission, the reduction of pathological impulses from the muscles to the central nervous system.

The third property of muscle relaxants is the prevention of muscular spasms during epileptic status, tetanus, rabies, etc. Note that the skeletal muscle of a man relaxes when taking muscle relaxant tablets, but amnesia and loss of consciousness are not comes.

Classification of muscle relaxants

Muscle relaxants are divided into 3 groups depending on the effect they have on the neuromuscular synapses:

• Non-depolarizing muscle relaxantsadditionally divided into drugs short (less than 20 minutes), medium (less than 40 minutes) and long-acting more than 40 minutes). Their mechanism of action is the effect of competitive neuromuscular blockers on the postsynaptic membrane. The ability to depolarize it is no longer due to the state of polarization. As a result, there is no contraction of the muscle fiber;
• Depolarizing muscle relaxants- preparations of ultrashort action (5-7 minutes). These include preparations of suxamethonium, which differ only in the salt included in the composition. The effect appears due to the depolarization of the postsynaptic membrane, the stimulation of the muscle fiber. But they do not leave the receptor instantly, therefore depolarization is short-lived, muscles quickly relax;
• Mixed preparations cause first a second and then a first block.

Side Effects of Muscle Relaxants

It is not recommended to start taking muscle relaxants yourself.

Be sure to consult a specialist to determine the exact cause of pain and the appointment of an integrated treatment.

Improperly selected medications to relax the muscles or incorrect dosage can cause the following side effects:

• Drowsiness;
• Heart rhythm disturbances, fluctuations in blood pressure;
• Muscle pain after surgery;
• Dry mouth;
• Problems with urination;
• Malignant hyperthermia (caused by depolarizing muscle relaxants);
• With an increased level of potassium in the blood, hyperkalemia may develop;
• Increased intraocular pressure;
• Fasciculation is a side effect of all depolarizing muscle relaxants.

Preparations for muscle relaxation

Consider the main drugs for relaxing the muscles of nondepolarizing and depolarizing action.

Decamethonium is a depolarizing muscle relaxant of powerful action. Also called decakuran, sinkuran, eulizin. The maximum action occurs in 3 minutes. To reduce the force of brush compression by 95% in an ordinary person it is enough, mg.

Dithilin is widely used in CIS countries as a muscle relaxant for short-term operations.

As a rule, it is administered intravenously. The effect occurs after 1 minute, the action time is from 5 to 10 minutes.

If administered intramuscularly, the effect develops in 2-4 minutes.

Atracurium. The second name is the tractor. Produced in ampoules by, and 5 ml. A representative of moderate muscle relaxants, recovery occurs in about 35 minutes.

Possible side effects in the form of skin hyperemia, anaphylactic reaction, lowering blood pressure, bronchospasm.

Most often, Atrakurium is used for surgical operations, intubation of the trachea.

Diplatcin refers to muscle relaxants of nondepolarizing action. The maximum action comes in 5-6 minutes and lasts from 18 to 25 minutes.

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Note that after restoring breathing, muscle relaxation still remains. With the introduction of large doses, an increase in blood pressure is possible.

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The disadvantages of the drug include individual intolerance.

Pipecuronium is a representative of long-lasting muscular relaxants. It is part of a group of nondepolarizing muscle relaxants. Also has the names arduan, arkuron. Possible side effects: hypotension, bradycardia, anaphylactic reaction.

Toxperin is one of the most powerful muscle relaxants of nondepolarizing action. It is a synthetic alkaloid of bottle curare.

Side effects are not noted, in addition, it can be used for allergic reactions.

Muscle relaxants with osteochondrosis

Tablets for muscle relaxation are often prescribed for osteochondrosis. Symptoms of this disease are reduced to dizziness, numbness, chest pain and lower back.

Often there is a spasm of the muscles of the back, the pain syndrome begins to progress because of muscle tension.

It is in this case that the appointment of muscle relaxants - tablets, which relax the skeletal muscles.

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Midsummer (tolperisone). One of the most popular drugs for relaxing the muscles of the neck and back with osteochondrosis, reflex syndrome therapy.

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It has the following actions: analgesic, vasodilating, myorelaxing. In addition, it perfectly combines with NSAIDs, increases mental ability, removes feelings of anxiety.

Numerous studies confirm the safety and good tolerability of the drug. After 1, an hour, patients notice a reduction in pain.

Contraindications to the admission of Midokalma is pregnancy, infant age, lactation period in women, individual intolerance.

Baclofen has the following advantages: relieves pain, muscle spasms increases the mobility of the spine, quickly absorbed into the digestive tract.

However, this drug has some side effects: nausea, dizziness, constipation, weakness. Therefore, the treatment of osteochondrosis with this muscle relaxant should be carried out exclusively under the supervision of a doctor.

With caution should be taken people suffering from diabetes, liver disease.

Affects the synapses of the medulla oblongata and spinal cord, therefore it is included in the group of muscle relaxants of the central action. The maximum effect comes in 4-6 minutes.

The advantages include a lack of influence on the liver, lobes and hemodynamics.

A source: http://www.sportobzor.ru/farmacevtika/myshechnye-relaksanty.html

The use of muscle relaxants to relieve muscle spasms

Miorelaxants for the removal of muscle spasms are prescribed for dislocation and surgical intervention, to combat cramps. After intake, they block impulses, promoting relaxation of the striated muscle.

Miorelaxants are used in the following fields of medicine:

• neurology - with complex therapy of osteochondrosis, arthritis;
• Surgery - to relax the muscles in the abdominal area;
• Diagnosis - to diagnose some pathologies.

Other causes of muscle relaxants:

• treatment of an electroconvulsive condition;
• anesthesia with partial stopping of the process of natural breathing;
• medicines of central influence (prophylaxis after trauma).

Acute pain that appears in the muscles causes a spasm. This limits the movement. Paralysis may occur. More often similar signs are observed at an osteochondrosis. Constant muscle spasms prevent their normal functioning, which requires long-term therapy.

To speed up the recovery, muscle relaxants are taken. They reduce inflammation, stopping pain. Relaxants are prescribed at any stage of osteochondrosis treatment. Preparations of the considered pharmacological group are not accepted in the following situations:

1. 1. Kidney pathology.
2. 2. Pregnancy.
3. 3. Lactation.
4. 4. Problems with the nervous system.
5. 5. Alcoholism.
6. 6. Ulcer.
7. 7. Children under 1 year of age.
8. 6. Ulcer.
9. 9. Epilepsy.

By the mechanism of influence on the body, muscle relaxants are classified into 2 types:

• peripheral drugs;
• central medicines.

The chemical composition is:

• glycerides (meprobamate);
• benzimidazoles - high efficiency has Flexen and Ketoprofen;
• mixed muscle relaxants (Sirdalud, Tolperizon).

Miorelaxants can act on the sick organism ultrashort, short, medium and long.

Peripheral agents effectively block the nerve impulses that come to the muscle fibers.

The reasons for their administration are associated with paralysis in tetanus, anesthesia, convulsions. Medicines of this category are classified into the following groups:

• Nondepolarizing (Arduan, Melliktin);
• depolarizing (Ditilin);
• mixed type (Dixonium).

During treatment, medications gently affect the cholinergic receptors of skeletal muscles, quickly relieving pain and spasms. Central muscle relaxants easily block synapses of muscle tissue. Monosynaptic reflexes are not affected. List of effective means of central impact:

1. 1. Baclofen.
2. 2. Tizanidine.
3. 3. Metacarbamol.

It is recommended to treat osteochondrosis in the thoracic, lumbar and cervical area under the supervision of a doctor. Miorelaxants are selected taking into account the manifested symptoms, the cause of the ailment, the patient's well-being.

Tablets, relaxing the muscle, take a certain rule. Therapy is performed in the unconscious state of the patient.

With the help of medicines, tension is removed, gas exchange is normalized, normal blood flow occurs.

If the drug is used for anesthesia, it is combined with an anesthetic.

Treatment of neurological pathologies associated with increased tone requires the use of muscle relaxant. Simultaneously, the drug relieves pain in the lower back and a crunch in the leg.

Miorelaxants are mandatory medications with intervertebral hernia.

But in some patients they can cause the following side reactions:

• the concentration of attention is lost;
• decreased blood pressure;
• increased nervous excitability;
• bed-wetting;
• gastrointestinal diseases;
• there are cramps.

Such effects occur if the patient takes the drug without following the prescribed dosage. More often this is observed when taking antisepolarizing drugs. In this case, you must stop treatment and consult a doctor.

To cure such conditions, a solution of Neostigmine is used. It is administered intravenously. Depolarizing muscle relaxants affect the body with a minimal negative effect.

To restore well-being, it is enough to stop taking them.

Rapid muscle relaxation is observed after taking the following muscle relaxants:

1. 1. Ditilina.
2. 2. Decamethony.

These medications are related to depolarizing agents. They have a powerful effect.

The maximum effect is observed at 3 minutes after taking a relatively small dose of medication.

Decamethonium is often used in surgery for short-term surgery.

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Imbretil is a mixed muscle relaxant that gives good results 3 minutes after intravenous injection. Medication Tracium is often used in the conduct of surgical intervention. Full recovery is observed 30 minutes after it was entered.

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Diplatcin is a nondepolarizing agent. Its effect is noticeable on the fifteenth minute after administration, and the duration of action is 20 minutes.

Medication Piperkuroniy is a nondepolarizing muscle relaxant that acts for 40 minutes. Another name is Arduan.

Medication Toxipherin is the most powerful non-depolarizing relaxant that is administered intravenously. Its effect is observed for 30-50 minutes.

With this disease appoint pills, relaxing skeletal muscles (Baclofen, Tolperizon).

The central muscle relaxant MI-301 acts 4 minutes after administration. Another name means - Reorgangan or Relaxil-G.

The drug Baclofen increases the mobility of the spine. It is well perceived by the body, quickly absorbed into the digestive tract. But Baclofen can provoke nausea, dizziness, constipation.

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The structure of the preparation is close to y-aminobutyric acid. Baclofen quickly binds to GABA receptors, effectively suppressing monosynaptic activity at the CM level.

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This provokes a decrease in muscle tone.

The drug Sirdalud effectively suppresses polysynaptic reflexes. For Sirdaluda a moderate central analgesic effect is characteristic. In this case, the patient may complain of dizziness, drowsiness.

The preparation is used for long-term therapy of compression and reflex complications, developed against the background of osteochondrosis, spondylosis.

The drug centrally affects the sick body, rapidly reducing muscle tone. Tolperisone effectively suppresses spinal cord reflex activity.

This drug is characterized by a slight vasodilator effect.

Medication Midokalm has an analgesic effect. Under its action, relaxed muscles are relaxed. After 60 minutes the pain decreases. The effectiveness of the drug is observed in the treatment of painful muscle spasms that are resistant to other types of treatment.

In this case, the pain is weakened after 90 minutes. Primary therapy lasts 1 week. With secondary therapy, the dosage of the drug increases.

Such a scheme of treatment helps to reduce pain, relieve anxiety, increase mental performance.

Plus, Midokalma is a good interaction with non-steroidal anti-inflammatory medication. This allows you to reduce the dosage of the last remedy, weakening or completely eliminating its adverse reactions. At the same time, the effectiveness of the current therapy remains.

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Midokalma lacks a sedative effect and muscle weakness. This advantage is proved in the course of various studies.

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Physicians distinguish various causes of the emergence of pathological conditions, for the elimination of which treatment with muscle relaxants is prescribed.

Before taking these drugs, it is recommended to consult a doctor. Since some of the drugs in this group are provoking side effects.

A source: http://spina-health.ru/miorelaksanty-dlya-snyatiya-myshechnyx-spazmov/

9 best muscle relaxants to relieve muscle spasms and back pain

Drugs that act as depressants of the central nervous system and have sedative and musculoskeletal relaxant properties are called muscle relaxants.

This list includes the names of active agents and medicines that are most effective.

Used in addition to rest, physiotherapy and other measures to relieve discomfort, muscle relaxants are useful for short-term use in acute painful conditions of the locomotor system apparatus.

Typically, muscle relaxants are prescribed in the early stages of back pain on a short-term basis to alleviate back pain associated with muscle spasms.

Muscle relaxants are also sometimes prescribed to patients with other symptoms of fibromyalgia. It is believed that they can alleviate the pain of tight muscles and muscle spasms that are common in this disease.

9 Most Effective Muscle Soothing Remedies

There are several types of muscle relaxants that are commonly used to treat back pain or neck pain.

Baclofen

Muscular insufficiency and muscle spasms, including those associated with spine traumas, are weakened with the help of baclofen. The medicine can be useful in the treatment of multiple sclerosis and stabbed neuralgia.

It is available in the form of tablets and can be consumed by children from the age of 12 years. Some common side effects may include nausea and vomiting, confusion, drowsiness, headache, or muscle weakness.

Chloroxazone

Chloroxoxazone is used to relieve discomfort from acute, painful sensations of the musculoskeletal system. It should not be used by patients with increased sensitivity to chlorosoxazone. The medicine can occasionally be toxic to the liver.

In case of loss of appetite, you should consult a doctor. Side effects include: nausea, vomiting, or fatigue; abdominal pain; dark urine; pale stools; yellowing of the skin or eyes. Chloroxoxazone is available as a tablet.

Not recommended for use during pregnancy.

Carisoprodol

Carisoprodolid relaxes muscles and relieves pain and stiffness caused by acute problems with bones and muscles that can be caused by trauma.

May be addictive, especially when used in combination with alcohol or other drugs that have sedative effects.

Patients with an anamnesis of acute intermittent porphyria or hypersensitivity to carbamate preparations, such as methocarbamol, should avoid carisoprodol. It is taken orally in the form of tablets and is also available in combination with aspirin or aspirin and codeine.

Cyclobenzaprine

Cyclobenzaprin relieves pain from muscle cramps and spasms.

It is not recommended for people with overactive thyroid gland, cardiac arrhythmia, heart failure or those who recently had a heart attack.

It can be used on a longer term basis and has a chemical structure associated with some antidepressants, although it is not an antidepressant.

Cyclobenzaprin is not approved for use in fibromyalgia, but it is sometimes useful in treating this condition. The drug is available in tablets and capsules. Cyclobenzaprin is the safest muscle relaxant for use during pregnancy.

Dantrolene

Dantrolen helps control chronic spasticity, including those associated with spinal injuries.

It is also used for conditions such as stroke, multiple sclerosis and cerebral palsy. Dantrolene is taken in the form of capsules.

Serious side effects are more likely in people with asthma, emphysema, bronchitis, or other lung diseases. May cause sensitization to light. Drowsiness is the most common side effect.

Diazepam (e.g., Valium)

This is an addition to the treatment of muscle spasms. Diazepam relieves symptoms of anxiety, including from refusal of alcohol and is used for epileptic seizures, such as epilepsy. Diazepam is usually limited to one to two weeks of use.

This restriction is due to its potential for habit formation and because it changes the sleep cycles, which leads to sleep difficulties after discontinuing the medication.

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Patients should also understand that diazepam is a depressant and can worsen the depression associated with chronic pain.

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Diazepam is not recommended for pregnant women, people suffering from myasthenia gravis, severe liver disease, sleep apnea (only oral tablets), serious breathing problems or some forms of glaucoma. It is marketed as a pill, liquid, injection and rectal gel.

Metaxalone (for example, Skelaxin, Metaxal)

Metaxalone directs pain and muscle spasms from stretching and muscle damage. Metaxalone in the smallest form causes relaxation of muscles from all muscle relaxants. Causes drowsiness.

It can be used in children aged 13 years and older with diseases of the musculoskeletal system, but it is not considered safe during pregnancy.

Metaxalone may affect the blood sugar level in people with diabetes. It is available in the form of a pill or injection.

Methocarbamol (e.g., Riboxin)

Methocarbamol relieves acute muscular pain. It is classified as carbamate and can also be used as an auxiliary therapy to control neuromuscular manifestations of tetanus, although it does not heal tetanus.

It can be taken in the form of tablets or by injection. Higher doses are sometimes prescribed in the first 48-72 hours of treatment. Those who have had an allergic reaction to any related drug should avoid taking methocarbamol.

Tizanidine (e.g., Zanaflex)

Muscular spasticity is controlled by tizanidine and is usually intended for daily activities and time, when the most important is the relief of spasticity.

It is used in adults with multiple sclerosis and spinal cord injury and in children with cerebral palsy.

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It should not be used by patients taking fluvoxamine or ciprofloxacin or people with liver disease.

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Those who have experienced an allergic reaction to tizanidine should also avoid taking this medication. It is available in the form of tablets and capsules, which are differently absorbed by the body when eating.

There is very little research on what type of muscle relaxant is more effective, so the choice of a particular medicine or its use is generally based on factors such as the patient's response to treatment and personal preferences, the possibility of abuse, possible drug interactions and side effects effects.

Medications are just one part of anesthesia. These drugs are designed to be one of the elements, usually on a short-term basis, of the overall strategy recovery, which goes beyond medicines, including rest, stretching, physical therapy and other exercises.

A source: https://okpozvonok.ru/lechenie/preparaty/9-luchshix-myshechnyx-relaksantov.html

Muscle relaxants for removing muscle cramps of the neck and legs: names, list, and how much they cost?

The muscle relaxants are a group of medications that have the ability to reduce the tone of the skeletal muscle with a decrease or complete restriction of movement.

What is muscle relaxants?

Qualitative muscle relaxants should reduce the excitability of muscle tissue, but do not suppress nerve impulses that support posture and give muscle strength during the movement.

Even with prolonged use of muscle relaxant will not have a big impact on the patient's activity and ability to work. Also, the drug should be combined with other drugs in the complex treatment of pathology.

There are two main groups of muscle relaxants:

1. depolarizing;
2. non-depolarizing.

Also there are drugs that have a central and peripheral effect.

Peripheral muscle relaxants are used:

Muscle relaxants of central action:

• do not affect the transmission of nerve impulses in the synapses;
• relieve muscle spasm.

Also, muscle relaxants are divided according to the duration of their action:

• too short, about 6 minutes;
• short to 20 minutes;
• average exposure to 35 minutes;
• long lasting up to 60 minutes.

With osteochondrosis

When osteochondrosis develops a steady development of the reflex tension of the muscles of the skeleton.

In the process of progression of the pathology pain syndrome appears, and the muscular spasm becomes more pronounced.

To eliminate this cause in the treatment of osteochondrosis in complex therapy, muscle relaxants are used.

Thanks to these tools, the following effects occur:

• muscle tension passes;
• decreases the pain threshold;
• the function of movement in the affected area is restored;
• to obtain a high result, it is necessary to take muscle relaxants for several weeks.

According to doctors, the most suitable muscle relaxants in the treatment of osteochondrosis are:

• Baclofen273 rubles for 50 tablets;
• Midokalmabout 510 rubles for 30 tablets;
• Sirdalud325 rubles for 30 tablets.

This group of funds in a short time can relieve muscle tension and eliminate pain. The muscle relaxants are indicated for oral administration, and their dose is selected individually for each patient.

This group of drugs is used in conjunction with nonsteroidal anti-inflammatory drugs, analgesics, gels of an irritating effect, and also in a complex with medical massage, medical gymnastics and manual therapy.

Contraindications

Only under the supervision of a specialist, it is recommended to take muscle relaxants.

They have a number of contraindications:

• renal and hepatic impairment;
• Parkinson's disease;
• stomach ulcer and duodenal ulcer;
• epilepsy;
• individual intolerance;
• the pathology of cerebral vessels.

Side effects:

• dizziness;
• weakness;
• nausea;
• intoxication;
• decrease in pressure;
• in rare cases, convulsions develop.

With neuralgia

Intercostal neuralgia is accompanied by pain in the chest due to nerve damage. If the treatment is not started at the time, the disease progresses rapidly and becomes chronic.

Therapeutic process in neuralgia is based on the use of drugs that will remove the symptoms and causes of the disease. In complex therapy with analgesics, non-steroidal anti-inflammatory drugs I prescribe muscle relaxants.

They will help to remove spasm of skeletal muscles, which are the main cause of neuralgia. The use of this group of drugs will help to get high results and quick recovery of the patient.

Doctors in neuralgia appoint the following muscle relaxants:

• Clonazepam is about 96 rubles;
• Tizanidine 147 rubles;
• Midokalm;
• Sirdalud.

Thanks to these agents, the effect on the affected and inflamed nerve is reduced and the pain syndrome is eliminated. The course of treatment depends on the severity of the disease and the individual characteristics of the patient's body.

The action of clonazepam in neuralgia:

• has a calming effect;
• anti-anxiety;
• anticonvulsant.

Contraindications:

• pathology of the liver and kidneys;
• fruit bearing;
• lactation;
• myasthenia gravis;
• joint administration with MAO inhibitors;
• it is not recommended to drive during the treatment;
• engage in work associated with increased danger and mental overexertion;
• you can not take alcohol.

Side effects:

• violation of coordination of movements;
• depression;
• increased excitability;
• nausea;
• fatigue.

With coxarthrosis

Coxarthrosis is a dystrophic lesion of the hip joint. If you start during treatment, you can suspend the process of destruction of the joint and restore its function.

The main task in the process of treatment of coxarthrosis is the removal of inflammation and pain syndrome. In combination with anti-inflammatory and analgesic agents, the patient is prescribed muscle relaxants.

They will help to relieve muscle tension and reduce pain syndrome.

Experts advise with coxarthrosis the following muscle relaxants:

• Tizalud about 195 rubles;
• Tolizor 200 rubles;
• Baclofen.

Action by Tizalud

Refers to muscle relaxants of central action.

Performs the following actions:

• stimulates the work of alpha-adrenergic receptors;
• reduces the transmission of nerve receptors in the spinal cord;
• restores muscle tone of the skeleton;
• gives a positive effect on muscle spasms;
• reduces the tone of the muscles of the skeleton during movement.

Contraindications:

• individual intolerance of components in the formulation;
• pathology of the kidneys and liver;
• pregnancy;
• lactation.

Side effects:

• nausea, vomiting;
• dizziness;
• increased pressure;
• tachycardia;
• jugular disorder of cerebral circulation;
• insomnia;
• a disruption in the work of the genitourinary system.

With sciatica

Sciatica is a lumbosacral radiculitis. Symptoms of the disease is pain, which spreads throughout the sciatic nerve.

The cause of the pathology is squeezing the roots of the spinal cord at the level of the lumbar region.

Read more about how to cure the sciatic nerve at home read here.

In most cases, sciatica affects patients after 35 years. To the development of the disease, there are a number of reasons that pathogenic microorganisms and bacteria secrete. A pain attack can last about 14 days.

Together with other drugs to relieve pain and inflammation, the patient is prescribed to undergo a medical course with muscle relaxants.

These drugs are used to eliminate reflex muscle spasm and to relieve pain.

In the beginning they can be used as injections, and then go to tablets. Dosage and duration of treatment depends on the severity of the disease and the individual characteristics of the patient.

Effective muscle relaxants in sciatica are:

• Carisoprodol is about 461 rubles;
• Diazepam 250 rubles;
• Sirdalud;
• Midsummer.

Application of Korysiprodol in Sciatica

Refers to muscle relaxants.

Its effect is due to the following factors:

• blocking of nerve impulses that are sent to the brain;
• together with physiotherapeutic methods gives a high result in the treatment of sciatica.

Contraindications:

• Porphyria;
• pathology of the liver and kidneys;
• pregnancy;
• lactation;
• children under 12 years.

Side effects:

• impaired vision;
• paralysis;
• development of allergic reactions;
• irritability;
• sleep disorders;
• depression;
• dizziness.

With bruxism

Bruxism is a pathology in which strong and involuntary compression of the upper and lower jaw occurs. The main manifestation of bruxism is the gnashing of teeth at night.

At the slightest sign of the disease, you need to contact the dentist.

After the examination, the doctor prescribes an additional examination and applies the method of treatment.

In addition to the appointment of dental technology, which will help to stop the process of erasing tooth enamel by applying tires, prosthetics, grinding.

Together with these technologies, drug treatment is added. These include muscle relaxants. Sometimes the doctor prescribes taking these medications immediately before bedtime. This will save muscle spasm and pain. This will help eliminate the creaking of teeth in a dream.

Effective in the treatment of bruxism are the following muscle relaxants:

• Fleksen 197 rubles;
• Isoprotan 250 rubles;
• Arduan 450 rubles;
• Detilin is 265 rubles.

Fleksen in the treatment of bruxism

Act:

• the membranes of lysosomes are restored;
• decreased activity of granulocytes;
• has anti-inflammatory effect;
• analgesic.

Contraindications:

• hypersensitivity;
• acute form of stomach disease;
• pregnancy;
• lactation;
• pathology of the liver and kidneys;
• of leukopenia.

Side effects:

• allergic reactions;
• hallucinations;
• decreased efficiency;
• lack of appetite;
• pressure reduction;
• tachycardia;
• bloating;
• nausea;
• sleep disturbance.

Feedback from specialists about muscle relaxants

Specialists in complex treatment necessarily prescribe to patients the intake of muscle relaxants. This group of drugs has proven itself in the treatment of osteochondrosis, bruxism, coxarthrosis, neuralgia and sciatica.

The main task of the remedies is to relieve unnecessary muscle tension and remove the pain syndrome, which is considered the main cause of the above pathologies.

Doctors in a particular disease apply various muscle relaxants, which have different effects on the body.

The disadvantage of this group of drugs is the rapid addiction and further dependence on them.

These funds, according to doctors, are forbidden to apply in childhood and adolescence. People who manage transport and have jobs related to increased concentration of attention and danger.

Like most drugs, muscle relaxants have their contraindications and side effects:

• increased drowsiness;
• apathy;
• migraine;
• nausea and vomiting;
• dizziness;
• muscle damage;
• pressure reduction;
• convulsions.

All these effects are typical for all types and groups of muscle relaxants. Specialists prescribe the dosage of the drug only in accordance with the severity of the pathological process and taking into account the individual characteristics of the organism.

Miorelaxants are well tolerated by patients and in rare cases can cause the development of allergic reactions. In case of overdose with muscle relaxants, it is necessary to urgently consult a doctor and undergo symptomatic treatment.

Means refer to new generation drugs and have a positive effect in the treatment of the musculoskeletal system, joints and other pathologies.

A source: http://SpinaSpina.com/lechenie/preparaty/miorelaksanty-dlya-snyatiya-spazmov.html

Scope of drugs - muscle relaxants

Muscle relaxants to relieve muscle spasms are drugs that help block neuromuscular impulses, relaxation of muscles, elimination of convulsions, are widely used in surgical practice.

General characteristics of muscle relaxants and their application

How will this or that muscle relaxant act on the body, depends on what its type is. In medicine, several types of this drug are called, which affects the decrease in muscle activity of the body.

Thus, central and peripheral muscle relaxants are isolated.

The main difference between these two groups is that the central muscle relaxants affect the muscular apparatus of the trunk as a whole, and the peripheral muscles affect the muscles of the local area.

The central group of such drugs include those that help to affect the neurons of the spinal cord, thereby helping to block their activity.

At the same time, central muscle relaxants do not affect monosynaptic reflexes, which is very convenient when used.

Central muscle relaxants have the following advantages:

• reduce muscle tone;
• relax the abdominal muscles;
• improve the quality of hardware diagnostics of pathologies;
• drugs that relieve muscle tension, are necessary for diseases that are accompanied by a violation of motor functions in the patient;
• drugs are used in the field of anaesthesiology;
• if there was a spasm in any part of the body, these drugs will come to the rescue.

The peripheral group of muscle relaxants influences the skeletal muscle holinoretseptors. For this reason, they are used for local elimination of muscle spasms. So, with the help of drugs, you can achieve relaxation of a small area of ​​the trunk, without effecting on other areas.

Peripheral drugs that can relieve muscle tension, are used in microsurgical surgery, with the direction of dislocation, in the treatment of stretching, for repositioning bone fragments.

In what cases is it forbidden to use drugs?

Such drugs do not have absolute contraindications to their use in the field of anesthesiology, except intolerance of the components. But there are relative contraindications, which are expressed in the following:

• in the presence of any lesion of the eyes;
• if a person suffers from a disease that is accompanied by an increase in intracranial pressure;
• if there is a severe burn;
• if a person suffers from a spinal cord disease;
• in the presence of congenital myotonia or muscular dystrophy;
• if there is a risk of developing such pathologies as arrhythmia and cardiac arrest;
• children;
• period of pregnancy.

Some of the drugs

If the doctor prescribes for a certain indication a medicine - muscle relaxant, then, as a rule, this is one of the following:

1. Baclofen. The drug helps suppress the hypertonic muscle, which is caused by a lesion of the spinal cord. The way of taking the medicine is oral, during the meal. Dosage is prescribed by the doctor individually. It is worth noting and side effects, which can be observed only when the dose is exceeded. These include: nausea, headache, muscle pain, tachycardia, diarrhea or constipation, an allergy to the skin (rash). It is forbidden to use Baclofen for individual intolerance to the drug, as well as during pregnancy and lactation.
2. Tizanidine (Sirdalud). Has a central effect on reducing muscle tone, helps reduce spasmodic reaction. Assign the drug for diseases of the spinal cord, stroke, multiple sclerosis, myelopathy. Side effects may include: malaise, dry mouth of mucous membranes, low blood pressure, dizziness. Dosage is determined by the doctor in each case individually.
3. Midsummer. The central effect agent is prescribed for admission in case of myelopathy, multiple sclerosis, spastic paralysis, spondylosis and spondyloarthrosis. Dosage is appointed by the attending physician in each case individually, taking into account the course of the disease and the tolerability of such a drug. Side effects are: headache, nausea and vomiting, low blood pressure, skin allergy (rash). Relative contraindications can be considered as periods of pregnancy and lactation.
4. Clonazepam. Assign with epilepsy, infantile spasms, hypertonic muscles, panic disorders. Contraindications are: the state of acute respiratory failure, severe depression, intolerance to the components of the drug, coma and shock. In pregnancy and lactation, the use of clonazepam is prohibited. If the dosage is exceeded, side effects may occur: fatigue and malaise, headache, nausea and vomiting, tachycardia, anemia.
5. Orfenadrine. Typically, this tool is prescribed for any injury to the muscles. Contraindications can be considered: intolerance of the components of the drug, heart and kidney disease, stomach ulcer. If the dosage is exceeded, the general condition may worsen, dizziness, vomiting and nausea, headache, skin allergy (rash). The dosage is determined by the attending physician.
6. Methocarbamol. Such a remedy is not prescribed to those people who are diagnosed with kidney failure, there are epileptic seizures, as well as during pregnancy, breast-feeding, children under 12 years. Side effects include constipation and diarrhea, darkening of urine, fainting, skin allergies (rash), nausea and vomiting, headache and malaise.

Miorelaxants with back pain

Almost every person has experienced pain in the lower back in his life, and in some cases, it becomes simply unbearable.

Even the strongest person, such a symptom can be unsettled and significantly affect his daily life.

How to relieve pain in this department? Eliminate such symptoms with the help of muscle relaxants.

To be a source of pain in the lumbar region can be a fixed lifestyle, which leads a person for many years, as well as diseases that contribute to the damage of intervertebral discs, the distortion the spine. As a rule, the pain arises from increasing, beginning in the lumbar zone, increasing with time.

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Pain in the lower back arises because of muscle spasms that squeeze blood vessels and nerve roots.

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As a result, there is a violation of blood supply in this department, which can lead to more serious diseases.

With the help of muscle relaxants it is possible to eliminate such muscle spasms, which, in turn, contributes to the restoration of impaired blood circulation and the removal of pain.

It should be noted right away that, unfortunately, muscle relaxants do not eliminate the root cause of pain in the lower back. Additional methods for treating the underlying cause are massage, manual therapy and physical education. Drugs with this effect will only increase the effectiveness of treatment.

As a rule, before the complex treatment to eliminate muscular spasm appoint a reception of muscle relaxants of central action. The optimal duration of treatment with these drugs is determined by the attending physician, based on the course of the pathology.

To achieve a lasting effect of muscle relaxants, they are recommended to use at least 6 months.

Consider the main drugs - muscle relaxants, which are used for back pain:

1. Baclofen has a very fast action. Immediately after the first intake, the normal functioning of the muscular system is restored, and the overall well-being of the person is improved.
2. Sirdalud affects the human body in a complex way, eliminating muscle spasms, anesthetizing, removing rare attacks in the lumbar region and chronic.
3. Mydocalm is the most common remedy for osteochondrosis. Thanks to such a drug, you can achieve that the muscle (muscles) relax, the vessels will expand, and the specific department will cease to hurt. Use both tablets and injections.

What kind of tool is suitable for this or that person, the doctor determines on the basis of the results of diagnosis, the frequency of seizures and the general condition of the body.

Miorelaxants are medicines that have a strong effect on the body.

This is why self-medication with these drugs is strictly prohibited!

A source: http://drpozvonkov.ru/lechenie/medikomentoznoe/tabulas-injections/sfera-primeneniya-preparatov-miorelaksantov.html